PDB Information

PDB5IH8
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Toward the Validation of Maternal Embryonic Leucine Zipper Kinase: Discovery, Optimization of Highly Potent and Selective Inhibitors, and Preliminary Biology Insight.
Toure, B.B., Giraldes, J., Smith, T., Sprague, E.R., Wang, Y., Mathieu, S., Chen, Z., Mishina, Y., Feng, Y., Yan-Neale, Y., Shakya, S., Chen, D., Meyer, M., Puleo, D., Brazell, J.T., Straub, C., Sage, D., Wright, K., Yuan, Y., Chen, X., Duca, J., Kim, S., Tian, L., Martin, E., Hurov, K., Shao, W.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2016-02-29
Resolution1.850
CATH Insert Date19 Jun, 2016

PDB Images (2)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 20 Jun, 2016 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q14680 MELK_HUMAN Homo sapiens Maternal embryonic leucine zipper kinase