PDB 5if1
PDB Information
| PDB | 5IF1 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | Conformational Adaption May Explain the Slow Dissociation Kinetics of Roniciclib (BAY 1000394), a Type I CDK Inhibitor with Kinetic Selectivity for CDK2 and CDK9.
Acs Chem.Biol.
|
| Header | Transferase |
| Released | 2016-02-25 |
| Resolution | 2.610 |
| CATH Insert Date | 08 May, 2016 |
PDB Images (13)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 09 May, 2016 | Chopped |
| B | 09 May, 2016 | Chopped |
| C | 09 May, 2016 | Chopped |
| D | 09 May, 2016 | Chopped |
CATH Domains (8)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5if1A01 | 18 Jul, 2016 | 3.30.200.20 | Assigned |
| 5if1A02 | 18 Jul, 2016 | 1.10.510.10 | Assigned |
| 5if1B01 | 17 Jul, 2016 | 1.10.472.10 | Assigned |
| 5if1B02 | 17 Jul, 2016 | 1.10.472.10 | Assigned |
| 5if1C01 | 18 Jul, 2016 | 3.30.200.20 | Assigned |
| 5if1C02 | 18 Jul, 2016 | 1.10.510.10 | Assigned |
| 5if1D01 | 18 Jul, 2016 | 1.10.472.10 | Assigned |
| 5if1D02 | 18 Jul, 2016 | 1.10.472.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P20248 | CCNA2_HUMAN | Homo sapiens | Cyclin-A2 |
| P20248 | CCNA2_HUMAN | Homo sapiens | Cyclin-A2 |
| P24941 | CDK2_HUMAN | Homo sapiens | Cyclin-dependent kinase 2 |
| P24941 | CDK2_HUMAN | Homo sapiens | Cyclin-dependent kinase 2 |
