PDB Information

PDB5IDN
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Structure-Based Optimization of Potent, Selective, and Orally Bioavailable CDK8 Inhibitors Discovered by High-Throughput Screening.
Czodrowski, P., Mallinger, A., Wienke, D., Esdar, C., Poschke, O., Busch, M., Rohdich, F., Eccles, S.A., Ortiz-Ruiz, M.J., Schneider, R., Raynaud, F.I., Clarke, P.A., Musil, D., Schwarz, D., Dale, T., Urbahns, K., Blagg, J., Schiemann, K.
J. Med. Chem.
HeaderTransferase
Released2016-02-24
Resolution2.260
CATH Insert Date25 Dec, 2016

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 26 Dec, 2016 Chopped
B 26 Dec, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5idnA01 29 Dec, 2016 3.30.200.20 Assigned
5idnA02 29 Dec, 2016 1.10.510.10 Assigned
5idnB01 29 Dec, 2016 1.10.472.10 Assigned
5idnB02 29 Dec, 2016 1.10.472.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P24863 CCNC_HUMAN Homo sapiens Cyclin-C
P49336 CDK8_HUMAN Homo sapiens Cyclin-dependent kinase 8