PDB 5idn
PDB Information
| PDB | 5IDN |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | Structure-Based Optimization of Potent, Selective, and Orally Bioavailable CDK8 Inhibitors Discovered by High-Throughput Screening.
J. Med. Chem.
|
| Header | Transferase |
| Released | 2016-02-24 |
| Resolution | 2.260 |
| CATH Insert Date | 25 Dec, 2016 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 26 Dec, 2016 | Chopped |
| B | 26 Dec, 2016 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5idnA01 | 29 Dec, 2016 | 3.30.200.20 | Assigned |
| 5idnA02 | 29 Dec, 2016 | 1.10.510.10 | Assigned |
| 5idnB01 | 29 Dec, 2016 | 1.10.472.10 | Assigned |
| 5idnB02 | 29 Dec, 2016 | 1.10.472.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P24863 | CCNC_HUMAN | Homo sapiens | Cyclin-C |
| P49336 | CDK8_HUMAN | Homo sapiens | Cyclin-dependent kinase 8 |
