PDB Information

PDB5I43
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Sugar-Based Arylsulfonamide Carboxylates as Selective and Water-Soluble Matrix Metalloproteinase-12 Inhibitors.
Nuti, E., Cuffaro, D., D'Andrea, F., Rosalia, L., Tepshi, L., Fabbi, M., Carbotti, G., Ferrini, S., Santamaria, S., Camodeca, C., Ciccone, L., Orlandini, E., Nencetti, S., Stura, E.A., Dive, V., Rossello, A.
Chemmedchem
HeaderHydrolase
Released2016-02-11
Resolution1.950
CATH Insert Date17 Jul, 2016

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 18 Jul, 2016 Chopped
B 18 Jul, 2016 Chopped
C 18 Jul, 2016 Chopped
D 18 Jul, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5i43A00 01 Sep, 2016 3.40.390.10 Assigned
5i43B00 01 Sep, 2016 3.40.390.10 Assigned
5i43C00 01 Sep, 2016 3.40.390.10 Assigned
5i43D00 01 Sep, 2016 3.40.390.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P39900 MMP12_HUMAN Homo sapiens Macrophage metalloelastase
P39900 MMP12_HUMAN Homo sapiens Macrophage metalloelastase
P39900 MMP12_HUMAN Homo sapiens Macrophage metalloelastase
P39900 MMP12_HUMAN Homo sapiens Macrophage metalloelastase