PDB Information

PDB5HU9
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery and characterization of a novel potent type II native and mutant BCR-ABL inhibitor (CHMFL-074) for Chronic Myeloid Leukemia (CML)
Liu, F., Wang, B., Wang, Q., Qi, Z., Chen, C., Kong, L.L., Chen, J.Y., Liu, X., Wang, A., Hu, C., Wang, W., Wang, H., Wu, F., Ruan, Y., Qi, S., Liu, J., Zou, F., Hu, Z., Wang, W., Wang, L., Zhang, S., Yun, C.H., Zhai, Z., Liu, J., Liu, Q.
Oncotarget
HeaderTransferase/Transferase Inhibitor
Released2016-01-27
Resolution1.530
CATH Insert Date07 Aug, 2016

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Aug, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5hu9A01 01 Sep, 2016 3.30.200.20 Assigned
5hu9A02 01 Sep, 2016 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P00519 ABL1_HUMAN Homo sapiens Tyrosine-protein kinase ABL1