PDB Information

PDB5HI7
MethodX-RAY DIFFRACTION
Host Organismunidentified baculovirus
Gene SourceHomo sapiens
Primary Citation
Structure-Based Design of a Novel SMYD3 Inhibitor that Bridges the SAM-and MEKK2-Binding Pockets.
Van Aller, G.S., Graves, A.P., Elkins, P.A., Bonnette, W.G., McDevitt, P.J., Zappacosta, F., Annan, R.S., Dean, T.W., Su, D.S., Carpenter, C.L., Mohammad, H.P., Kruger, R.G.
Structure
HeaderTransferase/Inhibitor
Released2016-01-11
Resolution2.150
CATH Insert Date10 Apr, 2016

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2016 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
5hi7A01 14 May, 2016 2.170.270.10 Assigned
5hi7A02 14 May, 2016 6.10.140.2220 Assigned
5hi7A03 14 May, 2016 1.10.220.160 Assigned
5hi7A04 14 May, 2016 1.25.40.970 Assigned
5hi7A05 14 May, 2016 1.25.40.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9H7B4 SMYD3_HUMAN Homo sapiens Histone-lysine N-methyltransferase SMYD3