PDB 5ha9
PDB Information
| PDB | 5HA9 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli K-12 |
| Gene Source | Homo sapiens |
| Primary Citation | Crystal structure-based discovery of a novel synthesized PARP1 inhibitor (OL-1) with apoptosis-inducing mechanisms in triple-negative breast cancer.
Sci Rep
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2015-12-30 |
| Resolution | 4.010 |
| CATH Insert Date | 10 Apr, 2016 |
PDB Images (3)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 11 Apr, 2016 | Rejected |
| B | 11 Apr, 2016 | Rejected |
CATH Domains (0)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P09874 | PARP1_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase 1 |
| P09874 | PARP1_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase 1 |
