PDB 5h6q
PDB Information
| PDB | 5H6Q |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Development and crystallographic evaluation of histone H3 peptide with N-terminal serine substitution as a potent inhibitor of lysine-specific demethylase 1.
Bioorg. Med. Chem.
|
| Header | Oxidoreductase/Transcription/Inhibitor |
| Released | 2016-11-14 |
| Resolution | 2.530 |
| CATH Insert Date | 07 May, 2017 |
PDB Images (8)
PDB Prints
PDB Chains (3)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 May, 2017 | Chopped |
| B | 08 May, 2017 | Chopped |
| C | 08 May, 2017 | Rejected |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5h6qA01 | 12 May, 2017 | 1.10.10.10 | Assigned |
| 5h6qA02 | 12 May, 2017 | Holding pen | |
| 5h6qA03 | 12 May, 2017 | 1.10.287.80 | Assigned |
| 5h6qB00 | 12 May, 2017 | 1.20.58.1880 | Assigned |
UniProtKB Entries (3)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O60341 | KDM1A_HUMAN | Homo sapiens | Lysine-specific histone demethylase 1A |
| P68431 | H31_HUMAN | Homo sapiens | Histone H3.1 |
| Q9UKL0 | RCOR1_HUMAN | Homo sapiens | REST corepressor 1 |
