PDB Information

PDB5H4J
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
TAS-114, a First-in-Class Dual dUTPase/DPD Inhibitor, Demonstrates Potential to Improve Therapeutic Efficacy of Fluoropyrimidine-Based Chemotherapy.
Yano, W., Yokogawa, T., Wakasa, T., Yamamura, K., Fujioka, A., Yoshisue, K., Matsushima, E., Miyahara, S., Miyakoshi, H., Taguchi, J., Chong, K.T., Takao, Y., Fukuoka, M., Matsuo, K.
Mol. Cancer Ther.
HeaderHydrolase/Hydrolase Inhibitor
Released2016-11-01
Resolution1.800
CATH Insert Date14 Nov, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5h4jA00 10 Dec, 2017 2.70.40.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P33316 DUT_HUMAN Homo sapiens Deoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial