PDB 5h21

PDB Information

PDB5H21
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Discovery of novel trimethoxy-ring BRD4 bromodomain inhibitors: AlphaScreen assay, crystallography and cell-based assay.
Chen, Z., Zhang, H., Liu, S., Xie, Y., Jiang, H., Lu, W., Xu, H., Yue, L., Zhang, Y., Ding, H., Zheng, M., Yu, K., Chen, K., Jiang, H., Luo, C.
Medchemcomm
HeaderPeptide Binding Protein/Inhibitor
Released2016-10-13
Resolution1.590
CATH Insert Date14 Nov, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5h21A01 10 Dec, 2017 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
CATH-Gene3D is a Global Biodata Core Resource Learn more...