PDB Information

PDB5H0B
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Activity cliff for 7-substituted pyrrolo-pyrimidine inhibitors of HCK explained in terms of predicted basicity of the amine nitrogen.
Yuki, H., Kikuzato, K., Koda, Y., Mikuni, J., Tomabechi, Y., Kukimoto-Niino, M., Tanaka, A., Shirai, F., Shirouzu, M., Koyama, H., Honma, T.
Bioorg. Med. Chem.
HeaderTransferase/Transferase Inhibitor
Released2016-10-04
Resolution1.650
CATH Insert Date14 Nov, 2017

PDB Images (2)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P08631 HCK_HUMAN Homo sapiens Tyrosine-protein kinase HCK