PDB 5fxr
PDB Information
| PDB | 5FXR |
| Method | X-RAY DIFFRACTION |
| Host Organism | ESCHERICHIA COLI |
| Gene Source | HOMO SAPIENS |
| Primary Citation | Discovery of a Potent, Selective, Orally Bioavailable, and Efficacious Novel 2-(Pyrazol-4-ylamino)-pyrimidine Inhibitor of the Insulin-like Growth Factor-1 Receptor (IGF-1R).
J. Med. Chem.
|
| Header | Transferase |
| Released | 2016-03-02 |
| Resolution | 2.400 |
| CATH Insert Date | 06 Nov, 2016 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 07 Nov, 2016 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5fxrA01 | 10 Nov, 2016 | 3.30.200.20 | Assigned |
| 5fxrA02 | 10 Nov, 2016 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P08069 | IGF1R_HUMAN | Homo sapiens | Insulin-like growth factor 1 receptor |
