PDB Information

PDB5FPF
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI BL21(DE3)
Gene SourceHOMO SAPIENS
Primary Citation
Design, Synthesis and Evaluation of Novel Dual- Binding Inhibitors of the Tankyrases and Wnt Signalling.
Nathubhai, A., Haikarainen, T., Hayward, P.C., Munoz-Descalzo, S., Tosh, D., Lloyd, M.D., Lehtio, L., Threadgill, M.D.
To be Published
HeaderTransferase
Released2015-11-30
Resolution2.600
CATH Insert Date25 Dec, 2016

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 26 Dec, 2016 Chopped
B 26 Dec, 2016 Chopped
C 26 Dec, 2016 Chopped
D 26 Dec, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5fpfA00 29 Dec, 2016 3.90.228.10 Assigned
5fpfB00 29 Dec, 2016 3.90.228.10 Assigned
5fpfC00 29 Dec, 2016 6.20.320.10 Assigned
5fpfD00 29 Dec, 2016 6.20.320.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2