PDB Information

PDB5FI6
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Design and evaluation of novel glutaminase inhibitors.
McDermott, L.A., Iyer, P., Vernetti, L., Rimer, S., Sun, J., Boby, M., Yang, T., Fioravanti, M., O'Neill, J., Wang, L., Drakes, D., Katt, W., Huang, Q., Cerione, R.
Bioorg.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2015-12-22
Resolution2.520
CATH Insert Date29 May, 2016

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 30 May, 2016 Chopped
B 30 May, 2016 Chopped
C 30 May, 2016 Chopped
D 30 May, 2016 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5fi6A01 16 Jul, 2016 1.10.238.210 Assigned
5fi6A02 16 Jul, 2016 3.40.710.10 Assigned
5fi6B01 16 Jul, 2016 1.10.238.210 Assigned
5fi6B02 16 Jul, 2016 3.40.710.10 Assigned
5fi6C01 16 Jul, 2016 1.10.238.210 Assigned
5fi6C02 16 Jul, 2016 3.40.710.10 Assigned
5fi6D01 16 Jul, 2016 1.10.238.210 Assigned
5fi6D02 16 Jul, 2016 3.40.710.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial
O94925 GLSK_HUMAN Homo sapiens Glutaminase kidney isoform, mitochondrial