PDB Information

PDB5EW3
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
A Novel Potent Oral Series of VEGFR2 Inhibitors Abrogate Tumor Growth by Inhibiting Angiogenesis.
Bold, G., Schnell, C., Furet, P., McSheehy, P., Bruggen, J., Mestan, J., Manley, P.W., Druckes, P., Burglin, M., Durler, U., Loretan, J., Reuter, R., Wartmann, M., Theuer, A., Bauer-Probst, B., Martiny-Baron, G., Allegrini, P., Goepfert, A., Wood, J., Littlewood-Evans, A.
J.Med.Chem.
HeaderTransferase
Released2015-11-20
Resolution2.500
CATH Insert Date27 Dec, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 28 Dec, 2015 Chopped
B 28 Dec, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5ew3A01 05 Jan, 2016 3.30.200.20 Assigned
5ew3A02 05 Jan, 2016 1.10.510.10 Assigned
5ew3B01 05 Jan, 2016 3.30.200.20 Assigned
5ew3B02 05 Jan, 2016 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P35968 VGFR2_HUMAN Homo sapiens Vascular endothelial growth factor receptor 2
P35968 VGFR2_HUMAN Homo sapiens Vascular endothelial growth factor receptor 2