PDB Information

PDB5ENP
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceEscherichia coli (strain K12)
Primary Citation
Molecular basis for inhibition of AcrB multidrug efflux pump by novel and powerful pyranopyridine derivatives.
Sjuts, H., Vargiu, A.V., Kwasny, S.M., Nguyen, S.T., Kim, H.S., Ding, X., Ornik, A.R., Ruggerone, P., Bowlin, T.L., Nikaido, H., Pos, K.M., Opperman, T.J.
Proc.Natl.Acad.Sci.USA
HeaderTransport Protein
Released2015-11-09
Resolution1.900
CATH Insert Date17 Apr, 2016

PDB Images (25)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
A 18 Apr, 2016 Chopped
B 18 Apr, 2016 Chopped
C 18 Apr, 2016 Chopped
D 18 Apr, 2016 Chopped
E 18 Apr, 2016 Chopped
F 18 Apr, 2016 Chopped

CATH Domains (18)

Domain ID Date inserted into CATH Superfamily CATH Status
5enpA01 09 Jan, 2018 3.30.70.1430 Assigned
5enpA02 09 Jan, 2018 3.30.70.1320 Assigned
5enpA03 09 Jan, 2018 Holding pen
5enpA04 09 Jan, 2018 3.30.70.1430 Assigned
5enpA05 09 Jan, 2018 3.30.70.1440 Assigned
5enpB01 09 Jan, 2018 3.30.70.1430 Assigned
5enpB02 09 Jan, 2018 3.30.70.1320 Assigned
5enpB03 09 Jan, 2018 Holding pen
5enpB04 09 Jan, 2018 3.30.70.1430 Assigned
5enpB05 09 Jan, 2018 3.30.70.1440 Assigned
5enpC01 09 Jan, 2018 3.30.70.1430 Assigned
5enpC02 09 Jan, 2018 3.30.70.1320 Assigned
5enpC03 09 Jan, 2018 Holding pen
5enpC04 09 Jan, 2018 3.30.70.1430 Assigned
5enpC05 09 Jan, 2018 3.30.70.1440 Assigned
5enpD00 30 Nov, 2016 1.25.40.20 Assigned
5enpE00 30 Nov, 2016 1.25.40.20 Assigned
5enpF00 30 Nov, 2016 1.25.40.20 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P31224 ACRB_ECOLI Escherichia coli K-12 Multidrug efflux pump subunit AcrB
P31224 ACRB_ECOLI Escherichia coli K-12 Multidrug efflux pump subunit AcrB
P31224 ACRB_ECOLI Escherichia coli K-12 Multidrug efflux pump subunit AcrB