PDB 5egu
PDB Information
| PDB | 5EGU |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21(DE3) |
| Gene Source | Homo sapiens |
| Primary Citation | Exploring Selective Inhibition of the First Bromodomain of the Human Bromodomain and Extra-terminal Domain (BET) Proteins.
J.Med.Chem.
|
| Header | Transcription |
| Released | 2015-10-27 |
| Resolution | 2.210 |
| CATH Insert Date | 10 Apr, 2016 |
PDB Images (9)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 11 Apr, 2016 | Chopped |
| B | 11 Apr, 2016 | Chopped |
| C | 11 Apr, 2016 | Chopped |
| D | 11 Apr, 2016 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5eguA01 | 08 May, 2016 | 1.20.920.10 | Assigned |
| 5eguB01 | 08 May, 2016 | 1.20.920.10 | Assigned |
| 5eguC01 | 08 May, 2016 | 1.20.920.10 | Assigned |
| 5eguD01 | 08 May, 2016 | 1.20.920.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
