PDB Information

PDB5E2R
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli 'BL21-Gold(DE3)pLysS AG'
Gene SourceHomo sapiens
Primary Citation
Discovery of 1,1'-Biphenyl-4-sulfonamides as a New Class of Potent and Selective Carbonic Anhydrase XIV Inhibitors.
La Regina, G., Coluccia, A., Famiglini, V., Pelliccia, S., Monti, L., Vullo, D., Nuti, E., Alterio, V., De Simone, G., Monti, S.M., Pan, P., Parkkila, S., Supuran, C.T., Rossello, A., Silvestri, R.
J.Med.Chem.
HeaderLyase
Released2015-10-01
Resolution1.600
CATH Insert Date15 Nov, 2015

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Nov, 2015 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5e2rA00 23 Nov, 2015 3.10.200.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P00918 CAH2_HUMAN Homo sapiens Carbonic anhydrase 2