PDB Information

PDB5E1E
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Identification of azabenzimidazoles as potent JAK1 selective inhibitors.
Vasbinder, M.M., Alimzhanov, M., Augustin, M., Bebernitz, G., Bell, K., Chuaqui, C., Deegan, T., Ferguson, A.D., Goodwin, K., Huszar, D., Kawatkar, A., Kawatkar, S., Read, J., Shi, J., Steinbacher, S., Steuber, H., Su, Q., Toader, D., Wang, H., Woessner, R., Wu, A., Ye, M., Zinda, M.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2015-09-29
Resolution2.300
CATH Insert Date06 Dec, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 07 Dec, 2015 Chopped
B 07 Dec, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5e1eA01 09 Dec, 2015 3.30.200.20 Assigned
5e1eA02 09 Dec, 2015 1.10.510.10 Assigned
5e1eB01 05 Jan, 2016 3.30.200.20 Assigned
5e1eB02 05 Jan, 2016 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P23458 JAK1_HUMAN Homo sapiens Tyrosine-protein kinase JAK1
P23458 JAK1_HUMAN Homo sapiens Tyrosine-protein kinase JAK1