PDB 5dw2
PDB Information
| PDB | 5DW2 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21(DE3) |
| Gene Source | Homo sapiens |
| Primary Citation | RVX-297- a novel BD2 selective inhibitor of BET bromodomains.
Biochem.Biophys.Res.Commun.
|
| Header | Protein Binding/Inhibitor |
| Released | 2015-09-22 |
| Resolution | 1.120 |
| CATH Insert Date | 17 Jul, 2016 |
PDB Images (3)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 18 Jul, 2016 | Chopped |
CATH Domains (1)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5dw2A01 | 01 Sep, 2016 | 1.20.920.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
