PDB 5dia
PDB Information
| PDB | 5DIA |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of 3,5-substituted 6-azaindazoles as potent pan-Pim inhibitors.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2015-08-31 |
| Resolution | 1.960 |
| CATH Insert Date | 08 Nov, 2015 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 09 Nov, 2015 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5diaA01 | 23 Nov, 2015 | 3.30.200.20 | Assigned |
| 5diaA02 | 23 Nov, 2015 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P11309 | PIM1_HUMAN | Homo sapiens | Serine/threonine-protein kinase pim-1 |
