PDB Information

PDB5CLS
MethodX-RAY DIFFRACTION
Host OrganismBaculovirus expression vector pFastBac1-HM
Gene SourceHomo sapiens
Primary Citation
Spiroepoxytriazoles Are Fumagillin-like Irreversible Inhibitors of MetAP2 with Potent Cellular Activity.
Morgen, M., Jost, C., Malz, M., Janowski, R., Niessing, D., Klein, C.D., Gunkel, N., Miller, A.K.
Acs Chem.Biol.
HeaderHydrolase
Released2015-07-16
Resolution1.750
CATH Insert Date17 Apr, 2016

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 18 Apr, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5clsA01 05 May, 2016 3.90.230.10 Assigned
5clsA02 05 May, 2016 1.10.10.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P50579 MAP2_HUMAN Homo sapiens Methionine aminopeptidase 2