PDB 5ax3
PDB Information
| PDB | 5AX3 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21 |
| Gene Source | Homo sapiens |
| Primary Citation | Identification of allosteric ERK2 inhibitors through in silico biased screening and competitive binding assay
Bioorg.Med.Chem.Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2015-07-14 |
| Resolution | 2.980 |
| CATH Insert Date | 10 Apr, 2016 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 11 Apr, 2016 | Chopped |
| B | 11 Apr, 2016 | Rejected |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5ax3A01 | 04 May, 2016 | 3.30.200.20 | Assigned |
| 5ax3A02 | 04 May, 2016 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P28482 | MK01_HUMAN | Homo sapiens | Mitogen-activated protein kinase 1 |
| P40763 | STAT3_HUMAN | Homo sapiens | Signal transducer and activator of transcription 3 |
