PDB Information

PDB5A81
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Structure-Based Optimization of Naphthyridones Into Potent Atad2 Bromodomain Inhibitors.
Bamborough, P., Chung, C., Furze, R.C., Grandi, P., Michon, A., Sheppard, R.J., Barnett, H., Diallo, H., Dixon, D.P., Douault, C., Jones, E.J., Karamshi, B., Mitchell, D.J., Prinjha, R.K., Rau, C., Watson, R.J., Werner, T., Demont, E.H.
J.Med.Chem.
HeaderHydrolase
Released2015-07-11
Resolution2.030
CATH Insert Date30 Aug, 2015

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 31 Aug, 2015 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5a81A00 03 Sep, 2015 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q6PL18 ATAD2_HUMAN Homo sapiens ATPase family AAA domain-containing protein 2