PDB Information

PDB4ZDK
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceMycobacterium tuberculosis (strain ATCC 25618 / H37Rv)
Primary Citation
Thiophenecarboxamide Derivatives Activated by EthA Kill Mycobacterium tuberculosis by Inhibiting the CTP Synthetase PyrG.
Mori, G., Chiarelli, L.R., Esposito, M., Makarov, V., Bellinzoni, M., Hartkoorn, R.C., Degiacomi, G., Boldrin, F., Ekins, S., de Jesus Lopes Ribeiro, A.L., Marino, L.B., Centarova, I., Svetlikova, Z., Blasko, J., Kazakova, E., Lepioshkin, A., Barilone, N., Zanoni, G., Porta, A., Fondi, M., Fani, R., Baulard, A.R., Mikusova, K., Alzari, P.M., Manganelli, R., de Carvalho, L.P., Riccardi, G., Cole, S.T., Pasca, M.R.
Chem.Biol.
HeaderLigase
Released2015-04-17
Resolution3.490
CATH Insert Date16 Aug, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 17 Aug, 2015 Chopped
B 17 Aug, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4zdkA01 24 Aug, 2015 3.40.50.300 Assigned
4zdkA02 24 Aug, 2015 3.40.50.880 Assigned
4zdkB01 24 Aug, 2015 3.40.50.300 Assigned
4zdkB02 24 Aug, 2015 3.40.50.880 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P9WHK7 PYRG_MYCTU Mycobacterium tuberculosis H37Rv CTP synthase
P9WHK7 PYRG_MYCTU Mycobacterium tuberculosis H37Rv CTP synthase