PDB Information

PDB4ZDI
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceMycobacterium tuberculosis (strain ATCC 25618 / H37Rv)
Primary Citation
Thiophenecarboxamide Derivatives Activated by EthA Kill Mycobacterium tuberculosis by Inhibiting the CTP Synthetase PyrG.
Mori, G., Chiarelli, L.R., Esposito, M., Makarov, V., Bellinzoni, M., Hartkoorn, R.C., Degiacomi, G., Boldrin, F., Ekins, S., de Jesus Lopes Ribeiro, A.L., Marino, L.B., Centarova, I., Svetlikova, Z., Blasko, J., Kazakova, E., Lepioshkin, A., Barilone, N., Zanoni, G., Porta, A., Fondi, M., Fani, R., Baulard, A.R., Mikusova, K., Alzari, P.M., Manganelli, R., de Carvalho, L.P., Riccardi, G., Cole, S.T., Pasca, M.R.
Chem.Biol.
HeaderLigase
Released2015-04-17
Resolution3.520
CATH Insert Date16 Aug, 2015

PDB Images (25)

PDB Prints

PDB Chains (8)

Chain ID Date inserted into CATH CATH Status
A 17 Aug, 2015 Chopped
B 17 Aug, 2015 Chopped
C 17 Aug, 2015 Chopped
D 17 Aug, 2015 Chopped
E 17 Aug, 2015 Chopped
F 17 Aug, 2015 Chopped
G 17 Aug, 2015 Chopped
H 17 Aug, 2015 Chopped

CATH Domains (16)

Domain ID Date inserted into CATH Superfamily CATH Status
4zdiA01 24 Aug, 2015 3.40.50.300 Assigned
4zdiA02 24 Aug, 2015 3.40.50.880 Assigned
4zdiB01 24 Aug, 2015 3.40.50.300 Assigned
4zdiB02 24 Aug, 2015 3.40.50.880 Assigned
4zdiC01 24 Aug, 2015 3.40.50.300 Assigned
4zdiC02 24 Aug, 2015 3.40.50.880 Assigned
4zdiD01 24 Aug, 2015 3.40.50.300 Assigned
4zdiD02 24 Aug, 2015 3.40.50.880 Assigned
4zdiE01 24 Aug, 2015 3.40.50.300 Assigned
4zdiE02 24 Aug, 2015 3.40.50.880 Assigned
4zdiF01 24 Aug, 2015 3.40.50.300 Assigned
4zdiF02 24 Aug, 2015 3.40.50.880 Assigned
4zdiG01 24 Aug, 2015 3.40.50.300 Assigned
4zdiG02 24 Aug, 2015 3.40.50.880 Assigned
4zdiH01 24 Aug, 2015 3.40.50.300 Assigned
4zdiH02 24 Aug, 2015 3.40.50.880 Assigned

UniProtKB Entries (8)

Accession Gene ID Taxon Description
P9WHK7 PYRG_MYCTU Mycobacterium tuberculosis H37Rv CTP synthase
P9WHK7 PYRG_MYCTU Mycobacterium tuberculosis H37Rv CTP synthase
P9WHK7 PYRG_MYCTU Mycobacterium tuberculosis H37Rv CTP synthase
P9WHK7 PYRG_MYCTU Mycobacterium tuberculosis H37Rv CTP synthase
P9WHK7 PYRG_MYCTU Mycobacterium tuberculosis H37Rv CTP synthase
P9WHK7 PYRG_MYCTU Mycobacterium tuberculosis H37Rv CTP synthase
P9WHK7 PYRG_MYCTU Mycobacterium tuberculosis H37Rv CTP synthase
P9WHK7 PYRG_MYCTU Mycobacterium tuberculosis H37Rv CTP synthase