PDB Information

PDB4Z6I
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
LP99: Discovery and Synthesis of the First Selective BRD7/9 Bromodomain Inhibitor.
Clark, P.G., Vieira, L.C., Tallant, C., Fedorov, O., Singleton, D.C., Rogers, C.M., Monteiro, O.P., Bennett, J.M., Baronio, R., Muller, S., Daniels, D.L., Mendez, J., Knapp, S., Brennan, P.E., Dixon, D.J.
Angew.Chem.Int.Ed.Engl.
HeaderTranscription
Released2015-04-05
Resolution1.950
CATH Insert Date28 Jun, 2015

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4z6iA00 27 Jul, 2015 1.20.920.10 Assigned
4z6iB00 27 Jul, 2015 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9H8M2 BRD9_HUMAN Homo sapiens Bromodomain-containing protein 9
Q9H8M2 BRD9_HUMAN Homo sapiens Bromodomain-containing protein 9