PDB Information

PDB4YHF
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Prolonged and tunable residence time using reversible covalent kinase inhibitors.
Bradshaw, J.M., McFarland, J.M., Paavilainen, V.O., Bisconte, A., Tam, D., Phan, V.T., Romanov, S., Finkle, D., Shu, J., Patel, V., Ton, T., Li, X., Loughhead, D.G., Nunn, P.A., Karr, D.E., Gerritsen, M.E., Funk, J.O., Owens, T.D., Verner, E., Brameld, K.A., Hill, R.J., Goldstein, D.M., Taunton, J.
Nat.Chem.Biol.
HeaderTransferase
Released2015-02-27
Resolution2.200
CATH Insert Date28 Jun, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4yhfA01 22 Jul, 2015 3.30.200.20 Assigned
4yhfA02 22 Jul, 2015 1.10.510.10 Assigned
4yhfB01 22 Jul, 2015 3.30.200.20 Assigned
4yhfB02 22 Jul, 2015 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q06187 BTK_HUMAN Homo sapiens Tyrosine-protein kinase BTK
Q06187 BTK_HUMAN Homo sapiens Tyrosine-protein kinase BTK