PDB Information

PDB4YFI
MethodX-RAY DIFFRACTION
Host Organismunidentified baculovirus
Gene SourceHomo sapiens
Primary Citation
Identification of Purines and 7-Deazapurines as Potent and Selective Type I Inhibitors of Troponin I-Interacting Kinase (TNNI3K).
Lawhorn, B.G., Philp, J., Zhao, Y., Louer, C., Hammond, M., Cheung, M., Fries, H., Graves, A.P., Shewchuk, L., Wang, L., Cottom, J.E., Qi, H., Zhao, H., Totoritis, R., Zhang, G., Schwartz, B., Li, H., Sweitzer, S., Holt, D.A., Gatto, G.J., Kallander, L.S.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2015-02-25
Resolution2.700
CATH Insert Date04 Oct, 2015

PDB Images (5)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 05 Oct, 2015 Holding pen
B 05 Oct, 2015 Holding pen
C 05 Oct, 2015 Domchop review
D 05 Oct, 2015 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q59H18 TNI3K_HUMAN Homo sapiens Serine/threonine-protein kinase TNNI3K
Q59H18 TNI3K_HUMAN Homo sapiens Serine/threonine-protein kinase TNNI3K
Q59H18 TNI3K_HUMAN Homo sapiens Serine/threonine-protein kinase TNNI3K
Q59H18 TNI3K_HUMAN Homo sapiens Serine/threonine-protein kinase TNNI3K