PDB Information

PDB4XJS
MethodX-RAY DIFFRACTION
Host OrganismPichia
Gene SourceHomo sapiens
Primary Citation
Discovery of 4-Amino-8-quinoline Carboxamides as Novel, Submicromolar Inhibitors of NAD-Hydrolyzing Enzyme CD38.
Becherer, J.D., Boros, E.E., Carpenter, T.Y., Cowan, D.J., Deaton, D.N., Haffner, C.D., Jeune, M.R., Kaldor, I.W., Poole, J.C., Preugschat, F., Rheault, T.R., Schulte, C.A., Shearer, B.G., Shearer, T.W., Shewchuk, L.M., Smalley, T.L., Stewart, E.L., Stuart, J.D., Ulrich, J.C.
J.Med.Chem.
HeaderHydrolase, Transferase
Released2015-01-09
Resolution2.800
CATH Insert Date06 Sep, 2015

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 07 Sep, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4xjsA01 11 Sep, 2015 1.20.82.10 Assigned
4xjsA02 11 Sep, 2015 3.40.50.720 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P28907 CD38_HUMAN Homo sapiens ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1