PDB Information

PDB4WA9
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Axitinib effectively inhibits BCR-ABL1(T315I) with a distinct binding conformation.
Pemovska, T., Johnson, E., Kontro, M., Repasky, G.A., Chen, J., Wells, P., Cronin, C.N., McTigue, M., Kallioniemi, O., Porkka, K., Murray, B.W., Wennerberg, K.
Nature
HeaderTransferase/Transferase Inhibitor
Released2014-08-28
Resolution2.200
CATH Insert Date28 Jun, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4wa9A01 15 Jul, 2015 3.30.200.20 Assigned
4wa9A02 15 Jul, 2015 1.10.510.10 Assigned
4wa9B01 15 Jul, 2015 3.30.200.20 Assigned
4wa9B02 15 Jul, 2015 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00519 ABL1_HUMAN Homo sapiens Tyrosine-protein kinase ABL1
P00519 ABL1_HUMAN Homo sapiens Tyrosine-protein kinase ABL1