PDB 4wa9
PDB Information
PDB | 4WA9 |
Method | X-RAY DIFFRACTION |
Host Organism | Spodoptera frugiperda |
Gene Source | Homo sapiens |
Primary Citation | Axitinib effectively inhibits BCR-ABL1(T315I) with a distinct binding conformation.
Nature
|
Header | Transferase/Transferase Inhibitor |
Released | 2014-08-28 |
Resolution | 2.200 |
CATH Insert Date | 28 Jun, 2015 |
PDB Images (7)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 29 Jun, 2015 | Chopped |
B | 29 Jun, 2015 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4wa9A01 | 15 Jul, 2015 | 3.30.200.20 | Assigned |
4wa9A02 | 15 Jul, 2015 | 1.10.510.10 | Assigned |
4wa9B01 | 15 Jul, 2015 | 3.30.200.20 | Assigned |
4wa9B02 | 15 Jul, 2015 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P00519 | ABL1_HUMAN | Homo sapiens | Tyrosine-protein kinase ABL1 |
P00519 | ABL1_HUMAN | Homo sapiens | Tyrosine-protein kinase ABL1 |