PDB Information

PDB4UQH
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceTRYPANOSOMA CRUZI
Primary Citation
4-Aminopyridyl-Based Cyp51 Inhibitors as Anti-Trypanosoma Cruzi Drug Leads with Improved Pharmacokinetic Profile and in Vivo Potency.
Calvet, C.M., Vieira, D.F., Choi, J.Y., Kellar, D., Cameron, M.D., Siqueira-Neto, J.L., Gut, J., Johnston, J.B., Lin, L., Khan, S., Mckerrow, J.H., Roush, W.R., Podust, L.M.
J.Med.Chem.
HeaderOxidoreductase
Released2014-06-23
Resolution2.430
CATH Insert Date24 Aug, 2014

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 25 Aug, 2014 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4uqhA00 29 Aug, 2014 1.10.630.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q7Z1V1 CP51_TRYCC Trypanosoma cruzi strain CL Brener Sterol 14-alpha demethylase