PDB 4u45
PDB Information
PDB | 4U45 |
Method | X-RAY DIFFRACTION |
Host Organism | Spodoptera frugiperda |
Gene Source | Homo sapiens |
Primary Citation | Fragment-based identification and optimization of a class of potent pyrrolo[2,1-f][1,2,4]triazine MAP4K4 inhibitors.
Bioorg.Med.Chem.Lett.
|
Header | Transferase/Transferase Inhibitor |
Released | 2014-07-23 |
Resolution | 2.580 |
CATH Insert Date | 14 Sep, 2014 |
PDB Images (7)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 15 Sep, 2014 | Chopped |
B | 15 Sep, 2014 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4u45A01 | 16 Sep, 2014 | 3.30.200.20 | Assigned |
4u45A02 | 16 Sep, 2014 | 1.10.510.10 | Assigned |
4u45B01 | 16 Sep, 2014 | 3.30.200.20 | Assigned |
4u45B02 | 16 Sep, 2014 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
O95819 | M4K4_HUMAN | Homo sapiens | Mitogen-activated protein kinase kinase kinase kinase 4 |
O95819 | M4K4_HUMAN | Homo sapiens | Mitogen-activated protein kinase kinase kinase kinase 4 |