PDB 4tpt
PDB Information
| PDB | 4TPT |
| Method | X-RAY DIFFRACTION |
| Host Organism | unidentified baculovirus |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of a Type III Inhibitor of LIM Kinase 2 That Binds in a DFG-Out Conformation.
Acs Med.Chem.Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2014-06-09 |
| Resolution | 2.600 |
| CATH Insert Date | 09 Nov, 2014 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 10 Nov, 2014 | Chopped |
| B | 10 Nov, 2014 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4tptA01 | 13 Nov, 2014 | 3.30.200.20 | Assigned |
| 4tptA02 | 13 Nov, 2014 | 1.10.510.10 | Assigned |
| 4tptB01 | 12 Nov, 2014 | 3.30.200.20 | Assigned |
| 4tptB02 | 12 Nov, 2014 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P53671 | LIMK2_HUMAN | Homo sapiens | LIM domain kinase 2 |
| P53671 | LIMK2_HUMAN | Homo sapiens | LIM domain kinase 2 |
