PDB Information

PDB4TK0
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Insights into the binding of PARP inhibitors to the catalytic domain of human tankyrase-2.
Qiu, W., Lam, R., Voytyuk, O., Romanov, V., Gordon, R., Gebremeskel, S., Vodsedalek, J., Thompson, C., Beletskaya, I., Battaile, K.P., Pai, E.F., Rottapel, R., Chirgadze, N.Y.
Acta Crystallogr.,Sect.D
HeaderTransferase
Released2014-05-25
Resolution1.650
CATH Insert Date16 Nov, 2014

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 17 Nov, 2014 Chopped
B 17 Nov, 2014 Chopped
C 17 Nov, 2014 Chopped
D 17 Nov, 2014 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4tk0A00 26 Nov, 2014 3.90.228.10 Assigned
4tk0B00 26 Nov, 2014 3.90.228.10 Assigned
4tk0C00 26 Nov, 2014 3.90.228.10 Assigned
4tk0D00 26 Nov, 2014 3.90.228.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2
Q9H2K2 TNKS2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase tankyrase-2