PDB Information

PDB4RZ8
MethodX-RAY DIFFRACTION
Host OrganismHomo Sapiens
Gene SourceHuman immunodeficiency virus 1
Primary Citation
Structure-Based Design of a Small Molecule CD4-Antagonist with Broad Spectrum Anti-HIV-1 Activity.
Curreli, F., Kwon, Y.D., Zhang, H., Scacalossi, D., Belov, D.S., Tikhonov, A.A., Andreev, I.A., Altieri, A., Kurkin, A.V., Kwong, P.D., Debnath, A.K.
J.Med.Chem.
HeaderViral Protein
Released2014-12-18
Resolution1.900
CATH Insert Date20 Sep, 2015

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 21 Sep, 2015 Chopped
B 21 Sep, 2015 Chopped
C 21 Sep, 2015 Chopped
D 21 Sep, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4rz8A01 13 Jul, 2016 2.170.40.20 Assigned
4rz8B01 13 Jul, 2016 2.170.40.20 Assigned
4rz8C01 13 Jul, 2016 2.170.40.20 Assigned
4rz8D01 13 Jul, 2016 2.170.40.20 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
A0A0M3KKW9 A0A0M3KKW9_9HIV1 Human immunodeficiency virus 1 clade A/E 93TH057 HIV-1 gp120 core
A0A0M3KKW9 A0A0M3KKW9_9HIV1 Human immunodeficiency virus 1 clade A/E 93TH057 HIV-1 gp120 core
A0A0M3KKW9 A0A0M3KKW9_9HIV1 Human immunodeficiency virus 1 clade A/E 93TH057 HIV-1 gp120 core
A0A0M3KKW9 A0A0M3KKW9_9HIV1 Human immunodeficiency virus 1 clade A/E 93TH057 HIV-1 gp120 core