PDB Information

PDB4RYD
MethodX-RAY DIFFRACTION
Host OrganismHomo sapiens
Gene SourceHomo sapiens
Primary Citation
Novel Furin Inhibitors with Potent Anti-infectious Activity.
Hardes, K., Becker, G.L., Lu, Y., Dahms, S.O., Kohler, S., Beyer, W., Sandvig, K., Yamamoto, H., Lindberg, I., Walz, L., von Messling, V., Than, M.E., Garten, W., Steinmetzer, T.
Chemmedchem
HeaderHydrolase/Hydrolase Inhibitor
Released2014-12-15
Resolution2.150
CATH Insert Date28 Jun, 2015

PDB Images (25)

PDB Prints

PDB Chains (12)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped
C 29 Jun, 2015 Chopped
D 29 Jun, 2015 Chopped
E 29 Jun, 2015 Chopped
F 29 Jun, 2015 Chopped
H 29 Jun, 2015 Rejected
I 29 Jun, 2015 Rejected
J 29 Jun, 2015 Rejected
K 29 Jun, 2015 Rejected
L 29 Jun, 2015 Rejected
N 29 Jun, 2015 Rejected

CATH Domains (12)

Domain ID Date inserted into CATH Superfamily CATH Status
4rydA01 10 Jul, 2015 3.40.50.200 Assigned
4rydA02 10 Jul, 2015 2.60.120.260 Assigned
4rydB01 10 Jul, 2015 3.40.50.200 Assigned
4rydB02 10 Jul, 2015 2.60.120.260 Assigned
4rydC01 10 Jul, 2015 3.40.50.200 Assigned
4rydC02 10 Jul, 2015 2.60.120.260 Assigned
4rydD01 10 Jul, 2015 3.40.50.200 Assigned
4rydD02 10 Jul, 2015 2.60.120.260 Assigned
4rydE01 10 Jul, 2015 3.40.50.200 Assigned
4rydE02 10 Jul, 2015 2.60.120.260 Assigned
4rydF01 10 Jul, 2015 3.40.50.200 Assigned
4rydF02 10 Jul, 2015 2.60.120.260 Assigned

UniProtKB Entries (6)

Accession Gene ID Taxon Description
P09958 FURIN_HUMAN Homo sapiens Furin
P09958 FURIN_HUMAN Homo sapiens Furin
P09958 FURIN_HUMAN Homo sapiens Furin
P09958 FURIN_HUMAN Homo sapiens Furin
P09958 FURIN_HUMAN Homo sapiens Furin
P09958 FURIN_HUMAN Homo sapiens Furin