PDB 4rvx
PDB Information
PDB | 4RVX |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Human immunodeficiency virus 1 |
Primary Citation | Enhanced antiviral activity by the P2-tris-tetrahydrofuran moiety of GRL-0519, a novel nonpeptidic HIV-1 protease inhibitor (PI), against multi-PI-resistant and highly darunavir-resistant strains of HIV-1.
To be Published
|
Header | Hydrolase/Hydrolase Inhibitor |
Released | 2014-11-28 |
Resolution | 1.960 |
CATH Insert Date | 15 May, 2016 |
PDB Images (9)
PDB Prints
PDB Chains (4)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 16 May, 2016 | Chopped |
B | 16 May, 2016 | Chopped |
C | 16 May, 2016 | Chopped |
D | 16 May, 2016 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4rvxA00 | 10 Jul, 2016 | 2.40.70.10 | Assigned |
4rvxB00 | 10 Jul, 2016 | 2.40.70.10 | Assigned |
4rvxC00 | 10 Jul, 2016 | 2.40.70.10 | Assigned |
4rvxD00 | 10 Jul, 2016 | 2.40.70.10 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q9J006 | Q9J006_9HIV1 | Human immunodeficiency virus 1 | Protease |
Q9J006 | Q9J006_9HIV1 | Human immunodeficiency virus 1 | Protease |
Q9J006 | Q9J006_9HIV1 | Human immunodeficiency virus 1 | Protease |
Q9J006 | Q9J006_9HIV1 | Human immunodeficiency virus 1 | Protease |