PDB Information

PDB4RVX
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHuman immunodeficiency virus 1
Primary Citation
Enhanced antiviral activity by the P2-tris-tetrahydrofuran moiety of GRL-0519, a novel nonpeptidic HIV-1 protease inhibitor (PI), against multi-PI-resistant and highly darunavir-resistant strains of HIV-1.
Yedidi, R.S., Maeda, K., Aoki, M., Garimella, H., Rao, K.V., Akasapu, S., Davis, D.A., Kaufman, J.D., Das, D., Wingfield, P.T., Amano, M., Ghosh, A.K., Mitsuya, H.
To be Published
HeaderHydrolase/Hydrolase Inhibitor
Released2014-11-28
Resolution1.960
CATH Insert Date15 May, 2016

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 16 May, 2016 Chopped
B 16 May, 2016 Chopped
C 16 May, 2016 Chopped
D 16 May, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4rvxA00 10 Jul, 2016 2.40.70.10 Assigned
4rvxB00 10 Jul, 2016 2.40.70.10 Assigned
4rvxC00 10 Jul, 2016 2.40.70.10 Assigned
4rvxD00 10 Jul, 2016 2.40.70.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q9J006 Q9J006_9HIV1 Human immunodeficiency virus 1 Protease
Q9J006 Q9J006_9HIV1 Human immunodeficiency virus 1 Protease
Q9J006 Q9J006_9HIV1 Human immunodeficiency virus 1 Protease
Q9J006 Q9J006_9HIV1 Human immunodeficiency virus 1 Protease