PDB Information

PDB4RRV
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
A small-molecule mimic of a peptide docking motif inhibits the protein kinase PDK1.
Rettenmaier, T.J., Sadowsky, J.D., Thomsen, N.D., Chen, S.C., Doak, A.K., Arkin, M.R., Wells, J.A.
Proc.Natl.Acad.Sci.USA
HeaderTransferase/Transferase Inhibitor
Released2014-11-06
Resolution1.410
CATH Insert Date28 Dec, 2014

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Dec, 2014 Chopped
B 29 Dec, 2014 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4rrvA01 06 Jan, 2015 3.30.200.20 Assigned
4rrvA02 06 Jan, 2015 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q16513 PKN2_HUMAN Homo sapiens Serine/threonine-protein kinase N2
O15530 PDPK1_HUMAN Homo sapiens 3-phosphoinositide-dependent protein kinase 1