PDB Information

PDB4RAK
MethodX-RAY DIFFRACTION
Host Organism
Gene SourceHomo sapiens
Primary Citation
Liver X Receptor (LXR) partial agonists: Biaryl pyrazoles and imidazoles displaying a preference for LXR beta.
Kick, E., Martin, R., Xie, Y., Flatt, B., Schweiger, E., Wang, T.L., Busch, B., Nyman, M., Gu, X.H., Yan, G., Wagner, B., Nanao, M., Nguyen, L., Stout, T., Plonowski, A., Schulman, I., Ostrowski, J., Kirchgessner, T., Wexler, R., Mohan, R.
Bioorg.Med.Chem.Lett.
HeaderTranscription/Agonist
Released2014-09-10
Resolution2.040
CATH Insert Date04 Jan, 2015

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Jan, 2015 Chopped
B 05 Jan, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4rakA00 20 Mar, 2016 1.10.565.10 Assigned
4rakB00 08 Jan, 2015 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P55055 NR1H2_HUMAN Homo sapiens Oxysterols receptor LXR-beta
P55055 NR1H2_HUMAN Homo sapiens Oxysterols receptor LXR-beta