PDB Information

PDB4R0I
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of O-(3-carbamimidoylphenyl)-l-serine amides as matriptase inhibitors using a fragment-linking approach
Goswami, R., Wohlfahrt, G., Mukherjee, S., Ghadiyaram, C., Nagaraj, J., Satyam, L.K., Subbarao, K., Gopinath, S., Krishnamurthy, N.R., Subramanya, H.S., Ramachandra, M.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2014-07-31
Resolution1.900
CATH Insert Date28 Jun, 2015

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4r0iA01 10 Jul, 2015 2.40.10.10 Assigned
4r0iA02 10 Jul, 2015 2.40.10.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9Y5Y6 ST14_HUMAN Homo sapiens Suppressor of tumorigenicity 14 protein
Q9Y5Y6 ST14_HUMAN Homo sapiens Suppressor of tumorigenicity 14 protein