PDB Information

PDB4QPS
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Tricyclic Covalent Inhibitors Selectively Target Jak3 through an Active Site Thiol.
Goedken, E.R., Argiriadi, M.A., Banach, D.L., Fiamengo, B.A., Foley, S.E., Frank, K.E., George, J.S., Harris, C.M., Hobson, A.D., Ihle, D.C., Marcotte, D., Merta, P.J., Michalak, M.E., Murdock, S.E., Tomlinson, M.J., Voss, J.W.
J.Biol.Chem.
HeaderTransferase/Transferase Inhibitor
Released2014-06-24
Resolution1.800
CATH Insert Date28 Jun, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
C 29 Jun, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4qpsA01 10 Jul, 2015 3.30.200.20 Assigned
4qpsA02 10 Jul, 2015 1.10.510.10 Assigned
4qpsC01 09 Jul, 2015 3.30.200.20 Assigned
4qpsC02 09 Jul, 2015 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P52333 JAK3_HUMAN Homo sapiens Tyrosine-protein kinase JAK3
P52333 JAK3_HUMAN Homo sapiens Tyrosine-protein kinase JAK3