PDB 4q1a
PDB Information
| PDB | 4Q1A |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Structure-guided development of deoxycytidine kinase inhibitors with nanomolar affinity and improved metabolic stability.
J.Med.Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2014-04-03 |
| Resolution | 1.900 |
| CATH Insert Date | 28 Jun, 2015 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 29 Jun, 2015 | Chopped |
| B | 29 Jun, 2015 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4q1aA00 | 09 Jul, 2015 | 3.40.50.300 | Assigned |
| 4q1aB00 | 10 Jul, 2015 | 3.40.50.300 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P27707 | DCK_HUMAN | Homo sapiens | Deoxycytidine kinase |
| P27707 | DCK_HUMAN | Homo sapiens | Deoxycytidine kinase |
