PDB 4py1
PDB Information
| PDB | 4PY1 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Kinase domain inhibition of leucine rich repeat kinase 2 (LRRK2) using a [1,2,4]triazolo[4,3-b]pyridazine scaffold.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase |
| Released | 2014-03-25 |
| Resolution | 2.160 |
| CATH Insert Date | 14 Sep, 2014 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 15 Sep, 2014 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4py1A01 | 16 Sep, 2014 | 3.30.200.20 | Assigned |
| 4py1A02 | 16 Sep, 2014 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P29597 | TYK2_HUMAN | Homo sapiens | Non-receptor tyrosine-protein kinase TYK2 |
