PDB Information

PDB4PX3
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery and Structure-Guided Optimization of Diarylmethanesulfonamide Disruptors of GK-GKRP Binding
Pennington, L.D., Bartberger, M.D., Croghan, M.D., Andrews, K.L., Ashton, K.S., Bourbeau, M.P., Chen, J., Chmait, S., Cupples, R., Fotsch, C.
To be Published
HeaderSugar Binding Protein/Inhibitor
Released2014-03-21
Resolution2.430
CATH Insert Date28 Jun, 2015

PDB Images (9)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
4px3A01 10 Jul, 2015 3.40.50.10490 Assigned
4px3A02 10 Jul, 2015 Holding pen
4px3A03 10 Jul, 2015 Holding pen
4px3B01 10 Jul, 2015 3.40.50.10490 Assigned
4px3B02 10 Jul, 2015 Holding pen
4px3B03 10 Jul, 2015 Holding pen

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q14397 GCKR_HUMAN Homo sapiens Glucokinase regulatory protein
Q14397 GCKR_HUMAN Homo sapiens Glucokinase regulatory protein