PDB Information

PDB4PI3
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceTrypanosoma cruzi
Primary Citation
Synthesis and Evaluation of Oxyguanidine Analogues of the Cysteine Protease Inhibitor WRR-483 against Cruzain.
Jones, B.D., Tochowicz, A., Tang, Y., Cameron, M.D., McCall, L.I., Hirata, K., Siqueira-Neto, J.L., Reed, S.L., McKerrow, J.H., Roush, W.R.
Acs Med.Chem.Lett.
HeaderHydrolase/Hydrolase Inhibitor
Released2014-05-08
Resolution1.270
CATH Insert Date30 Nov, 2014

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 01 Dec, 2014 Chopped
B 01 Dec, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4pi3A00 03 Dec, 2014 3.90.70.10 Assigned
4pi3B00 20 Mar, 2016 3.90.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P25779 CYSP_TRYCR Trypanosoma cruzi Cruzipain
P25779 CYSP_TRYCR Trypanosoma cruzi Cruzipain