PDB 4pci
PDB Information
| PDB | 4PCI |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of BRD4 bromodomain inhibitors by fragment-based high-throughput docking.
Bioorg.Med.Chem.Lett.
|
| Header | Transcription/Transcription Inhibitor |
| Released | 2014-04-15 |
| Resolution | 1.250 |
| CATH Insert Date | 18 May, 2014 |
PDB Images (3)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 19 May, 2014 | Chopped |
CATH Domains (1)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4pciA01 | 21 May, 2014 | 1.20.920.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
