PDB Information

PDB4P58
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMus musculus
Primary Citation
A fragment-based approach to identifying S-adenosyl-l-methionine -competitive inhibitors of catechol O-methyl transferase (COMT).
Lanier, M., Ambrus, G., Cole, D.C., Davenport, R., Ellery, J., Fosbeary, R., Jennings, A.J., Kadotani, A., Kamada, Y., Kamran, R., Matsumoto, S., Mizukami, A., Okubo, S., Okada, K., Saikatendu, K., Walsh, L., Wu, H., Hixon, M.S.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2014-03-15
Resolution2.060
CATH Insert Date06 Jul, 2014

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 07 Jul, 2014 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4p58A00 27 Oct, 2014 3.40.50.150 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O88587 COMT_MOUSE Mus musculus Catechol O-methyltransferase