PDB Information

PDB4NZ2
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-based ligand design to overcome CYP inhibition in drug discovery projects.
Branden, G., Sjogren, T., Schnecke, V., Xue, Y.
Drug Discov Today
HeaderOxidoreductase/Oxidoreductase Inhibitor
Released2013-12-11
Resolution2.450
CATH Insert Date24 Aug, 2014

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 25 Aug, 2014 Chopped
B 25 Aug, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4nz2A00 29 Aug, 2014 1.10.630.10 Assigned
4nz2B00 29 Aug, 2014 1.10.630.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P11712 CP2C9_HUMAN Homo sapiens Cytochrome P450 2C9
P11712 CP2C9_HUMAN Homo sapiens Cytochrome P450 2C9