PDB Information

PDB4NW5
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
2-Amino-7-substituted benzoxazole analogs as potent RSK2 inhibitors.
Costales, A., Mathur, M., Ramurthy, S., Lan, J., Subramanian, S., Jain, R., Atallah, G., Setti, L., Lindvall, M., Appleton, B.A., Ornelas, E., Feucht, P., Warne, B., Doyle, L., Basham, S.E., Aronchik, I., Jefferson, A.B., Shafer, C.M.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2013-12-05
Resolution1.940
CATH Insert Date23 Feb, 2014

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 24 Feb, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4nw5A01 07 Mar, 2014 3.30.200.20 Assigned
4nw5A02 07 Mar, 2014 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P51812 KS6A3_HUMAN Homo sapiens Ribosomal protein S6 kinase alpha-3